scholarly journals Scaffold hopping of fused piperidine-type NK3 receptor antagonists to reduce environmental impact

2019 ◽  
Vol 27 (10) ◽  
pp. 2019-2026 ◽  
Author(s):  
Koki Yamamoto ◽  
Shinsuke Inuki ◽  
Hiroaki Ohno ◽  
Shinya Oishi
Keyword(s):  
Environmental Impact ◽  
Scaffold Hopping ◽  
Receptor Antagonists ◽  
Nk3 Receptor

Development of novel NK3 receptor antagonists with reduced environmental impact

2016 ◽  
Vol 24 (16) ◽  
pp. 3494-3500 ◽  
Author(s):  
Koki Yamamoto ◽  
Shiho Okazaki ◽  
Hiroaki Ohno ◽  
Fuko Matsuda ◽  
Satoshi Ohkura ◽  
...  
Keyword(s):  
Environmental Impact ◽  
Receptor Antagonists ◽  
Nk3 Receptor

NK3 receptor antagonists: the next generation of antipsychotics?

2005 ◽  
Vol 4 (12) ◽  
pp. 967-975 ◽  
Author(s):  
Will Spooren ◽  
Claus Riemer ◽  
Herbert Meltzer
Keyword(s):  
Next Generation ◽  
Receptor Antagonists ◽  
Nk3 Receptor

MAPPING THE BINDING SITE FOR TACHYKININ NK3 RECEPTOR ANTAGONISTS

2008 ◽  
Vol 102 (1-3) ◽  
pp. 65 ◽  
Author(s):  
Pari Malherbe ◽  
Caterina Bissantz ◽  
Frédéric Knoflach ◽  
Maria-Clemencia Hernandez ◽  
Lucinda Steward ◽  
...  
Keyword(s):  
Binding Site ◽  
Receptor Antagonists ◽  
Nk3 Receptor

Identification of a new series of non-peptidic NK3 receptor antagonists

2011 ◽  
Vol 21 (5) ◽  
pp. 1498-1501 ◽  
Author(s):  
Karsten Juhl ◽  
Tore Hansen ◽  
Jan Kehler ◽  
Nikolay A. Khanzhin ◽  
Morten B. Nørgaard ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Nk3 Receptor

scholarly journals In vitro and in vivo characterization of NK3 receptors in the rabbit eye by use of selective non-peptide NK3 receptor antagonists

1997 ◽  
Vol 122 (3) ◽  
pp. 469-476 ◽  
Author(s):  
Andrew D. Medhurst ◽  
Douglas W. P. Hay ◽  
Andrew A. Parsons ◽  
Lenox D. Martin ◽  
Don E. Griswold
Keyword(s):  
Receptor Antagonists ◽  
Rabbit Eye ◽  
Nk3 Receptor ◽  
In Vivo Characterization

Discovery of a novel indole series of EP1 receptor antagonists by scaffold hopping

2008 ◽  
Vol 18 (8) ◽  
pp. 2684-2690 ◽  
Author(s):  
Adrian Hall ◽  
Andy Billinton ◽  
Susan H. Brown ◽  
Anita Chowdhury ◽  
Gerard M.P. Giblin ◽  
...  
Keyword(s):  
Scaffold Hopping ◽  
Receptor Antagonists ◽  
Ep1 Receptor ◽  
Indole Series

N′,2-Diphenylquinoline-4-carbohydrazide based NK3 receptor antagonists II

2006 ◽  
Vol 16 (22) ◽  
pp. 5752-5756 ◽  
Author(s):  
Jason M. Elliott ◽  
Robert W. Carling ◽  
Gary G. Chicchi ◽  
James Crawforth ◽  
Peter H. Hutson ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Nk3 Receptor
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