Design, synthesis, and biological evaluation of α-hydroxyacyl-AMS inhibitors of amino acid adenylation enzymes

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2016.09.027 ◽

2016 ◽

Vol 26 (21) ◽

pp. 5340-5345 ◽

Author(s):

Tony D. Davis ◽

Poornima Mohandas ◽

Maria I. Chiriac ◽

Glennon V. Bythrow ◽

Luis E.N. Quadri ◽

...

Keyword(s):

Biological Evaluation ◽

Design Synthesis ◽

Synthesis And Biological Evaluation

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Design, synthesis and biological evaluation of novel tripeptidyl epoxyketone derivatives constructed from β-amino acid as proteasome inhibitors

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2014.04.011 ◽

2014 ◽

Vol 22 (11) ◽

pp. 2955-2965 ◽

Author(s):

Jiankang Zhang ◽

Jiayi Cao ◽

Lei Xu ◽

Yubo Zhou ◽

Tao Liu ◽

...

Keyword(s):

Proteasome Inhibitors ◽

Biological Evaluation ◽

Design Synthesis ◽

Synthesis And Biological Evaluation

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Design, synthesis, and biological evaluation of water-soluble amino acid prodrug conjugates derived from combretastatin, dihydronaphthalene, and benzosuberene-based parent vascular disrupting agents

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2016.01.007 ◽

2016 ◽

Vol 24 (5) ◽

pp. 938-956 ◽

Author(s):

Laxman Devkota ◽

Chen-Ming Lin ◽

Tracy E. Strecker ◽

Yifan Wang ◽

Justin K. Tidmore ◽

...

Keyword(s):

Biological Evaluation ◽

Water Soluble ◽

Vascular Disrupting Agents ◽

Design Synthesis ◽

Synthesis And Biological Evaluation ◽

Vascular Disrupting

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Design, synthesis, and biological evaluation of novel 4-anilinoquinazoline derivatives bearing amino acid moiety as potential EGFR kinase inhibitors

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2017.02.061 ◽

2017 ◽

Vol 130 ◽

pp. 393-405 ◽

Author(s):

You-Guang Zheng ◽

Jun Su ◽

Cai-Yun Gao ◽

Ping Jiang ◽

Lin An ◽

...

Keyword(s):

Kinase Inhibitors ◽

Biological Evaluation ◽

Acid Moiety ◽

Design Synthesis ◽

Amino Acid Moiety ◽

Synthesis And Biological Evaluation ◽

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Design, synthesis and biological evaluation of novel amino acid ureido derivatives as aminopeptidase N/CD13 inhibitors

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2012.04.035 ◽

2012 ◽

Vol 20 (12) ◽

pp. 3807-3815 ◽

Author(s):

Li Su ◽

Yuping Jia ◽

Lei Zhang ◽

Yingying Xu ◽

Hao Fang ◽

...

Keyword(s):

Biological Evaluation ◽

Aminopeptidase N ◽

Design Synthesis ◽

Synthesis And Biological Evaluation

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Design, synthesis, and biological evaluation of ligustrazine - betulin amino-acid/dipeptide derivatives as anti-tumor agents

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2019.111839 ◽

2020 ◽

Vol 185 ◽

pp. 111839

Author(s):

Wen-Bo Guo ◽

Hao Zhang ◽

Wen-Qiang Yan ◽

Yi-Man Liu ◽

Fei Zhou ◽

...

Keyword(s):

Biological Evaluation ◽

Design Synthesis ◽

Synthesis And Biological Evaluation

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Design, synthesis, and biological evaluation of a dansyled amino acid derivative as an imaging agent for apoptosis

Tetrahedron Letters ◽

10.1016/j.tetlet.2008.08.091 ◽

2008 ◽

Vol 49 (45) ◽

pp. 6429-6432 ◽

Author(s):

Wenbin Zeng ◽

Weimin Miao ◽

George Kabalka ◽

Michael Le Puil ◽

John Biggerstaff ◽

...

Keyword(s):

Acid Derivative ◽

Biological Evaluation ◽

Imaging Agent ◽

Amino Acid Derivative ◽

Design Synthesis ◽

Synthesis And Biological Evaluation

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Design, Synthesis, and Biological Evaluation of a Novel Water-soluble Prodrug of Docetaxel with Amino Acid as a Linker

Chemical Biology & Drug Design ◽

10.1111/cbdd.12762 ◽

2016 ◽

Vol 88 (3) ◽

pp. 363-369 ◽

Author(s):

Huan Ma ◽

Gang Chen ◽

Tao Wang ◽

Qingeng Li ◽

Yan Liu

Keyword(s):

Biological Evaluation ◽

Water Soluble ◽

Design Synthesis ◽

Synthesis And Biological Evaluation

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Targeting species specific amino acid residues: Design, synthesis and biological evaluation of 6-substituted pyrrolo[2,3-d]pyrimidines as dihydrofolate reductase inhibitors and potential anti-opportunistic infection agents

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2018.04.032 ◽

2018 ◽

Vol 26 (9) ◽

pp. 2640-2650 ◽

Author(s):

Khushbu Shah ◽

Xin Lin ◽

Sherry F. Queener ◽

Vivian Cody ◽

Jim Pace ◽

...

Keyword(s):

Dihydrofolate Reductase ◽

Biological Evaluation ◽

Amino Acid Residues ◽

Design Synthesis ◽

Specific Amino Acid ◽

Reductase Inhibitors ◽

Species Specific ◽

Synthesis And Biological Evaluation ◽

Dihydrofolate Reductase Inhibitors

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Design, synthesis and biological evaluation of novel 31-hexyloxy chlorin e6-based 152- or 131-amino acid derivatives as potent photosensitizers for photodynamic therapy

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2020.112715 ◽

2020 ◽

Vol 207 ◽

pp. 112715

Author(s):

Xing-Jie Zhang ◽

Gui-Yan Han ◽

Chang-Yong Guo ◽

Zhi-Qiang Ma ◽

Mei-Yu Lin ◽

...

Keyword(s):

Photodynamic Therapy ◽

Biological Evaluation ◽

Amino Acid Derivatives ◽

Design Synthesis ◽

Synthesis And Biological Evaluation

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Design, Synthesis and Biological Evaluation of some Chalcone Derivatives as Potential Pancreatic Lipase Inhibitors

10.3390/ecsoc-17-b024 ◽

2013 ◽

Author(s):

Dao Tran

Keyword(s):

Pancreatic Lipase ◽

Biological Evaluation ◽

Design Synthesis ◽

Chalcone Derivatives ◽

Pancreatic Lipase Inhibitors ◽

Synthesis And Biological Evaluation

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