Synthesis of cis and trans 4-amido 2-carboxytetrahydroquinolines, high affinity ligands at the glycine site of the NMDA receptor

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/s0960-894x(00)80148-1 ◽

1992 ◽

Vol 2 (5) ◽

pp. 371-374 ◽

Author(s):

Graeme I. Stevenson ◽

Paul D. Leeson ◽

Michael Rowley ◽

Ian Sanderson ◽

Ian Stansfield

Keyword(s):

Nmda Receptor ◽

Glycine Site ◽

Affinity Ligands ◽

High Affinity ◽

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Requirements for high affinity binding of glycine analogs to the glycine site of the NMDA receptor complex

European Journal of Pharmacology Molecular Pharmacology ◽

10.1016/0922-4106(93)90131-r ◽

1993 ◽

Vol 247 (1) ◽

pp. 1-10 ◽

Author(s):

Anita H. Lewin ◽

Phil Skolnick ◽

Juan Carlos Marvizon ◽

Ian A. Paul ◽

J.Phillip Bowen

Keyword(s):

Nmda Receptor ◽

Affinity Binding ◽

Receptor Complex ◽

Glycine Site ◽

High Affinity Binding ◽

High Affinity ◽

Nmda Receptor Complex

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Effects of L-701,324, a high-affinity antagonist at the N-methyl-D-aspartate (NMDA) receptor glycine site, on the rat electroencephalogram

Naunyn-Schmiedeberg s Archives of Pharmacology ◽

10.1007/pl00005013 ◽

1997 ◽

Vol 355 (6) ◽

pp. 779-786 ◽

Author(s):

T. P. Obrenovitch ◽

Aidan M. Hardy ◽

Elias Zilkha

Keyword(s):

Nmda Receptor ◽

Glycine Site ◽

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Faculty Opinions recommendation of Discovering high-affinity ligands for proteins: SAR by NMR.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1087717.541807 ◽

2007 ◽

Author(s):

Robert Powers

Keyword(s):

Affinity Ligands ◽

High Affinity ◽

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Infectious bronchitis virus: Identification of Gallus gallus APN high-affinity ligands with antiviral effects

Antiviral Research ◽

10.1016/j.antiviral.2020.104998 ◽

2021 ◽

Vol 186 ◽

pp. 104998

Author(s):

Xiaoqi Sun ◽

Lanlan Li ◽

Long Pan ◽

Zheng Wang ◽

Huijie Chen ◽

...

Keyword(s):

Infectious Bronchitis Virus ◽

Gallus Gallus ◽

Affinity Ligands ◽

Virus Identification ◽

Infectious Bronchitis ◽

High Affinity ◽

Antiviral Effects

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Purification of bacterial virulence factor pertactin using high affinity ligands

Biochemical Engineering Journal ◽

10.1016/j.bej.2020.107760 ◽

2020 ◽

Vol 164 ◽

pp. 107760

Author(s):

Umatheny Umatheva ◽

Braden Sweeting ◽

Léo Sauvaget ◽

Nerissa Dela Rosa ◽

John Riley ◽

...

Keyword(s):

Virulence Factor ◽

Bacterial Virulence ◽

Affinity Ligands ◽

High Affinity ◽

Bacterial Virulence Factor

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Synthesis and biological evaluation of 6-aryl-6 H -pyrrolo[3,4- d ]pyridazine derivatives as high-affinity ligands of the α 2 δ subunit of voltage-gated calcium channels

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2004.02.070 ◽

2004 ◽

Vol 14 (9) ◽

pp. 2031-2034 ◽

Author(s):

Tao Hu ◽

Brian A Stearns ◽

Brian T Campbell ◽

Jeannie M Arruda ◽

Chixu Chen ◽

...

Keyword(s):

Calcium Channels ◽

Biological Evaluation ◽

Affinity Ligands ◽

Voltage Gated ◽

High Affinity ◽

Voltage Gated Calcium Channels ◽

Pyridazine Derivatives ◽

Synthesis And Biological Evaluation

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Identification of Elf-1 and B61 as high affinity ligands for the receptor tyrosine kinase MDK1

Oncogene ◽

10.1038/sj.onc.1200800 ◽

1997 ◽

Vol 14 (1) ◽

pp. 35-43 ◽

Author(s):

Thomas Ciossek ◽

Axel Ullrich

Keyword(s):

Tyrosine Kinase ◽

Receptor Tyrosine Kinase ◽

Affinity Ligands ◽

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High Throughput Screening of High-Affinity Ligands for Proteins with Anion-Binding Sites using Desorption Electrospray Ionization (DESI) Mass Spectrometry

Journal of the American Society for Mass Spectrometry ◽

10.1007/s13361-013-0753-3 ◽

2014 ◽

Vol 25 (3) ◽

pp. 454-463 ◽

Author(s):

Xin Lu ◽

Baoming Ning ◽

Dacheng He ◽

Lingyun Huang ◽

Xiangjun Yue ◽

...

Keyword(s):

Mass Spectrometry ◽

Electrospray Ionization ◽

High Throughput ◽

Binding Sites ◽

High Throughput Screening ◽

Desorption Electrospray Ionization ◽

Anion Binding ◽

Affinity Ligands ◽

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Interaction among NMDA receptor-, NMDA glycine site- and AMPA receptor antagonists in spinally mediated analgesia

Canadian Journal of Anesthesia/Journal canadien d anesthésie ◽

10.1007/bf03019004 ◽

2000 ◽

Vol 47 (7) ◽

pp. 693-698 ◽

Author(s):

Tomoki Nishiyama

Keyword(s):

Nmda Receptor ◽

Ampa Receptor ◽

Glycine Site ◽

Receptor Antagonists

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Chiral Auxiliary Mediated Conjugate Reduction and Asymmetric Protonation: Synthesis of High Affinity Ligands for HIV Protease Inhibitors

The Journal of Organic Chemistry ◽

10.1021/jo00124a042 ◽

1995 ◽

Vol 60 (19) ◽

pp. 6198-6201 ◽

Author(s):

Arun K. Ghosh ◽

Wenming Liu

Keyword(s):

Protease Inhibitors ◽

Chiral Auxiliary ◽

Hiv Protease ◽

Hiv Protease Inhibitors ◽

Affinity Ligands ◽

High Affinity ◽

Conjugate Reduction

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