5-Hydroxytryptamine1A Receptor Occupancy by Novel Full Antagonist 2-[4-[4-(7-Chloro-2,3-dihydro-1,4-benzdioxyn-5-yl)-1-piperazinyl]butyl]-1,2-benzisothiazol-3-(2H)-one-1,1-dioxide: A [11C][O-methyl-3H]-N-(2-(4-(2-methoxyphenyl)-1-piperazinyl)ethyl)-N-(2-pyridinyl)cyclohexanecarboxamide Trihydrochloride (WAY-100635) Positron Emission Tomography Study in Humans

Receptor Occupancy ◽

Emission Tomography ◽

Positron Emission ◽

Way 100635

Correction to: An open-label, positron emission tomography study of the striatal D2/D3 receptor occupancy and pharmacokinetics of single-dose oral brexpiprazole in healthy participants

European Journal of Clinical Pharmacology ◽

10.1007/s00228-020-03071-z ◽

2021 ◽

Author(s):

Dean F. Wong ◽

Arash Raoufinia ◽

Patricia Bricmont ◽

James R. Brašić ◽

Robert D. McQuade ◽

...

Keyword(s):

Single Dose ◽

Receptor Occupancy ◽

Emission Tomography ◽

D3 Receptor ◽

Open Label ◽

Positron Emission ◽

Dose Oral ◽

Healthy Participants

A Positron Emission Tomography Study of Quetiapine in Schizophrenia: A Preliminary Finding of an Antipsychotic Effect With Only Transiently High Dopamine D2 Receptor Occupancy

Archives of General Psychiatry ◽

10.1001/archpsyc.57.6.553 ◽

2000 ◽

Vol 57 (6) ◽

pp. 553-559 ◽

Cited By ~ 253

Author(s):

S. Kapur

Keyword(s):

Dopamine D2 Receptor ◽

D2 Receptor ◽

Preliminary Finding ◽

Receptor Occupancy ◽

Emission Tomography ◽

Dopamine D2 Receptor Occupancy ◽

Antipsychotic Effect ◽

Dopamine D2 receptor occupancy by perospirone: a positron emission tomography study in patients with schizophrenia and healthy subjects

Psychopharmacology ◽

10.1007/s00213-010-1783-1 ◽

2010 ◽

Vol 209 (4) ◽

pp. 285-290 ◽

Cited By ~ 7

Author(s):

Ryosuke Arakawa ◽

Hiroshi Ito ◽

Akihiro Takano ◽

Masaki Okumura ◽

Hidehiko Takahashi ◽

...

Keyword(s):

Healthy Subjects ◽

Dopamine D2 Receptor ◽

D2 Receptor ◽

Receptor Occupancy ◽

Emission Tomography ◽

Dopamine D2 ◽

Dopamine D2 Receptor Occupancy ◽

Histamine H1 receptor occupancy by the new-generation antipsychotics olanzapine and quetiapine: a positron emission tomography study in healthy volunteers

Psychopharmacology ◽

10.1007/s00213-015-4002-2 ◽

2015 ◽

Vol 232 (19) ◽

pp. 3497-3505 ◽

Cited By ~ 13

Author(s):

Hirotoshi Sato ◽

Chihiro Ito ◽

Kotaro Hiraoka ◽

Manabu Tashiro ◽

Katsuhiko Shibuya ◽

...

Keyword(s):

Healthy Volunteers ◽

Receptor Occupancy ◽

Emission Tomography ◽

H1 Receptor ◽

Histamine H1 Receptor ◽

Positron Emission ◽

New Generation ◽

Histamine H1 Receptor Occupancy

Striatal and extrastriatal dopamine D2 receptor occupancy by the partial agonist antipsychotic drug aripiprazole in the human brain: a positron emission tomography study with [11C]raclopride and [11C]FLB457

Psychopharmacology ◽

10.1007/s00213-011-2633-5 ◽

2012 ◽

Vol 222 (1) ◽

pp. 165-172 ◽

Cited By ~ 10

Author(s):

Keisuke Takahata ◽

Hiroshi Ito ◽

Harumasa Takano ◽

Ryosuke Arakawa ◽

Hironobu Fujiwara ◽

...

Keyword(s):

Human Brain ◽

Antipsychotic Drug ◽

Dopamine D2 Receptor ◽

Partial Agonist ◽

D2 Receptor ◽

Receptor Occupancy ◽

Emission Tomography ◽

A positron emission tomography study in healthy volunteers to estimate mGluR5 receptor occupancy of AZD2066 — Estimating occupancy in the absence of a reference region

NeuroImage ◽

10.1016/j.neuroimage.2013.05.006 ◽

2013 ◽

Vol 82 ◽

pp. 160-169 ◽

Cited By ~ 30

Author(s):

Matts Kågedal ◽

Zsolt Cselényi ◽

Svante Nyberg ◽

Patrick Raboisson ◽

Lars Ståhle ◽

...

Keyword(s):

Healthy Volunteers ◽

Receptor Occupancy ◽

Emission Tomography ◽

Reference Region ◽

Dopamine D2 receptor occupancy of lumateperone (ITI-007): a Positron Emission Tomography Study in patients with schizophrenia

Neuropsychopharmacology ◽

10.1038/s41386-018-0251-1 ◽

2018 ◽

Vol 44 (3) ◽

pp. 598-605 ◽

Cited By ~ 8

Author(s):

Kimberly E. Vanover ◽

Robert E. Davis ◽

Yun Zhou ◽

Weiguo Ye ◽

James R. Brašić ◽

...

Keyword(s):

Dopamine D2 Receptor ◽

D2 Receptor ◽

Receptor Occupancy ◽

Emission Tomography ◽

Dopamine D2 ◽

Dopamine D2 Receptor Occupancy ◽

Brain 5-HT 2A receptor occupancy of deramciclane in humans after a single oral administration - a positron emission tomography study

Psychopharmacology ◽

10.1007/s002130051034 ◽

1999 ◽

Vol 145 (1) ◽

pp. 76-81 ◽

Cited By ~ 6

Author(s):

H. Kanerva ◽

Harry Vilkman ◽

Kjell Någren ◽

Olavi Kilkku ◽

Mikko Kuoppamäki ◽

...

Keyword(s):

Oral Administration ◽

Receptor Occupancy ◽

Emission Tomography ◽

Positron Emission ◽

Single Oral Administration

Histamine H1 receptor occupancy by the new-generation antidepressants fluvoxamine and mirtazapine: a positron emission tomography study in healthy volunteers

Psychopharmacology ◽

10.1007/s00213-013-3146-1 ◽

2013 ◽

Vol 230 (2) ◽

pp. 227-234 ◽

Cited By ~ 12

Author(s):

Hirotoshi Sato ◽

Chihiro Ito ◽

Manabu Tashiro ◽

Kotaro Hiraoka ◽

Katsuhiko Shibuya ◽

...

Keyword(s):

Healthy Volunteers ◽

Receptor Occupancy ◽

Emission Tomography ◽

H1 Receptor ◽

Histamine H1 Receptor ◽

Positron Emission ◽

New Generation ◽

Histamine H1 Receptor Occupancy

An in vivo Positron Emission Tomography Study of Adenosine 2A Receptor Occupancy by Preladenant using 11C-SCH442416 in Healthy Subjects

Journal of Diagnostic Imaging in Therapy ◽

10.17229/jdit.2014-0712-002 ◽

2014 ◽

Vol 1 (1) ◽

pp. 20-48 ◽

Cited By ~ 2

Author(s):

Igor Grachev ◽

Miroslava Doder ◽

David Brooks ◽

Rainer Hinz

Keyword(s):

Healthy Subjects ◽

Receptor Occupancy ◽

Emission Tomography ◽

Positron Emission ◽

Adenosine 2A Receptor