scholarly journals Structure-activity relationship in piericidins inhibitors on the electron transport system in mitochondria.

1980 ◽  
Vol 44 (12) ◽  
pp. 2921-2924 ◽  
Author(s):  
Shigeo YOSHIDA ◽  
Yuichiro NAGAO ◽  
Akio WATANABE ◽  
Nobutaka TAKAHASHI
Keyword(s):  
Electron Transport ◽  
Transport System ◽  
Structure Activity Relationship ◽  
Electron Transport System ◽  
Activity Relationship ◽  
Structure Activity

Quantitative Structure Activity Relationship of Diphenylamines as Inhibitors of Photosynthetic Electron Transport and Photophosphorylation

1979 ◽  
Vol 34 (11) ◽  
pp. 1024-1027 ◽  
Author(s):  
Walter Oettmeier
Keyword(s):  
Electron Transport ◽  
Electron Flow ◽  
Photosynthetic Electron Transport ◽  
Quantitative Structure Activity Relationship ◽  
Structure Activity Relationship ◽  
Activity Relationship ◽  
Quantitative Structure ◽  
Structure Activity ◽  
Cyclic Photophosphorylation ◽  
Relationship Of

Abstract A number of 16 substituted diphenylamines have been tested for their inhibitory activity on photosynthetic NADP reduction and photophosphorylation. The most active compounds exhibited pI50 values of 6.0 in photosynthetic electron transport and 6.8 in cyclic photophosphorylation, respectively. The inhibition site in electron flow of the diphenylamines is located between the two photosystems. Necessary for high activity is the substitution of the phenyl moieties by several strongly electron withdrawing substituents. A quantitative structure activity relationship according to a parabolic Hansch approach could be accomplished by using the Hammett electronic parameter as the only variable.

Structure-activity relationship of (-) mammea A/BB derivatives against Leishmania amazonensis

Planta Medica ◽  
2008 ◽  
Vol 74 (09) ◽  
Author(s):  
MA Brenzan ◽  
CV Nakamura ◽  
BPD Filho ◽  
T Ueda-Nakamura ◽  
MCM Young ◽  
...  
Keyword(s):  
Structure Activity Relationship ◽  
Leishmania Amazonensis ◽  
Activity Relationship ◽  
Structure Activity ◽  
Relationship Of
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