N-Terminal Anthranoyl-Phenylalanine Derivatives as CCK1 Receptor Antagonists: The Final Approach

2005 ◽  
Vol 1 (5) ◽  
pp. 501-517 ◽  
Author(s):  
A. Varnavas ◽  
L. Lassiani ◽  
V. Valenta ◽  
A. Ciogli ◽  
F. Gasparrini ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Cck1 Receptor ◽  
Final Approach

Pyrazole CCK1 receptor antagonists

2007 ◽  
Vol 12 (11-12) ◽  
pp. 496-496
Author(s):  
P EDWARDS
Keyword(s):  
Receptor Antagonists ◽  
Cck1 Receptor

Pyrazole CCK1 receptor antagonists. Part 1: Solution-phase library synthesis and determination of Free–Wilson additivity

2006 ◽  
Vol 16 (1) ◽  
pp. 72-76 ◽  
Author(s):  
Kelly McClure ◽  
Michael Hack ◽  
Liming Huang ◽  
Clark Sehon ◽  
Magda Morton ◽  
...  
Keyword(s):  
Solution Phase ◽  
Library Synthesis ◽  
Receptor Antagonists ◽  
Cck1 Receptor

Pyrazole CCK1 receptor antagonists. Part 2: SAR studies by solid-phase library synthesis and determination of Free–Wilson additivity

2006 ◽  
Vol 16 (1) ◽  
pp. 77-80 ◽  
Author(s):  
Clark Sehon ◽  
Kelly McClure ◽  
Michael Hack ◽  
Magda Morton ◽  
Laurent Gomez ◽  
...  
Keyword(s):  
Solid Phase ◽  
Library Synthesis ◽  
Receptor Antagonists ◽  
Sar Studies ◽  
Cck1 Receptor

2D-QSAR and 3D-QSAR/CoMFA analyses of the N-terminal substituted anthranilic acid based CCK1 receptor antagonists: ‘Hic Rhodus, hic saltus’

2009 ◽  
Vol 17 (14) ◽  
pp. 5198-5206 ◽  
Author(s):  
Dimitra Hadjipavlou-Litina ◽  
Paolo Braiuca ◽  
Lucia Lassiani ◽  
Michela V. Pavan ◽  
Antonio Varnavas
Keyword(s):  
Anthranilic Acid ◽  
3D Qsar ◽  
Receptor Antagonists ◽  
2D Qsar ◽  
Cck1 Receptor

Anthranilic acid based CCK1 receptor antagonists: preliminary investigation on their second “touch point”

2005 ◽  
Vol 40 (6) ◽  
pp. 563-581 ◽  
Author(s):  
Antonio Varnavas ◽  
Lucia Lassiani ◽  
Valentina Valenta ◽  
Laura Mennuni ◽  
Francesco Makovec ◽  
...  
Keyword(s):  
Anthranilic Acid ◽  
Preliminary Investigation ◽  
Receptor Antagonists ◽  
Cck1 Receptor ◽  
Touch Point

Anthranilic acid derivatives: a new class of non-peptide CCK1 receptor antagonists

2003 ◽  
Vol 11 (5) ◽  
pp. 741-751 ◽  
Author(s):  
Antonio Varnavas ◽  
Lucia Lassiani ◽  
Valentina Valenta ◽  
Federico Berti ◽  
Laura Mennuni ◽  
...  
Keyword(s):  
Anthranilic Acid ◽  
Receptor Antagonists ◽  
New Class ◽  
Cck1 Receptor ◽  
Anthranilic Acid Derivatives

Anthranilic acid based CCK1 receptor antagonists: Blocking the receptor with the same ‘words’ of the endogenous ligand

2009 ◽  
Vol 17 (6) ◽  
pp. 2336-2350 ◽  
Author(s):  
Lucia Lassiani ◽  
Michela V. Pavan ◽  
Federico Berti ◽  
George Kokotos ◽  
Theodoros Markidis ◽  
...  
Keyword(s):  
Anthranilic Acid ◽  
Endogenous Ligand ◽  
Receptor Antagonists ◽  
Cck1 Receptor

SAR studies of 1,5-diarylpyrazole-based CCK1 receptor antagonists

2007 ◽  
Vol 17 (23) ◽  
pp. 6493-6498 ◽  
Author(s):  
Laurent Gomez ◽  
Michael D. Hack ◽  
Kelly McClure ◽  
Clark Sehon ◽  
Liming Huang ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Sar Studies ◽  
Cck1 Receptor
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