Crystallization of human leukocyte elastase with its inhibitor Pro44-eglin c

Dirk W. Heinz; Manfred Liersch; Markus G. Grütter

doi:10.1016/0022-2836(89)90474-9

Crystallization of human leukocyte elastase with its inhibitor Pro44-eglin c

Journal of Molecular Biology ◽

10.1016/0022-2836(89)90474-9 ◽

1989 ◽

Vol 207 (3) ◽

pp. 641-642 ◽

Cited By ~ 3

Author(s):

Dirk W. Heinz ◽

Manfred Liersch ◽

Markus G. Grütter

Keyword(s):

Human Leukocyte ◽

Leukocyte Elastase ◽

Human Leukocyte Elastase ◽

Eglin C

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Amino acids and peptides. Part 31. Total synthesis of eglin c. Part 1. Synthesis of a triacontapeptide corresponding to the C-terminal sequence 41–70 of eglin c and related peptides and studies on the relationship between the structure and inhibitory activity against human leukocyte elastase, csthepsin G and α-chymotrypsin

Journal of the Chemical Society Perkin Transactions 1 ◽

10.1039/p19910003315 ◽

1991 ◽

pp. 3315-3319 ◽

Cited By ~ 4

Author(s):

Yoshio Okada ◽

Satoshi Tsuboi

Keyword(s):

Amino Acids ◽

Total Synthesis ◽

Inhibitory Activity ◽

Human Leukocyte ◽

Terminal Sequence ◽

Leukocyte Elastase ◽

Human Leukocyte Elastase ◽

Eglin C ◽

The Relationship

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Amino acids and peptides. Part 32. Total synthesis of eglin c. Part 2. Synthesis of a heptacontapeptide corresponding to the entire amino acid sequence of eglin c and of related peptides, and studies on the relationship between the structure and inhibitory activity against human leukocyte elastase, cathepsin G and α-chymotrypsin

Journal of the Chemical Society Perkin Transactions 1 ◽

10.1039/p19910003321 ◽

1991 ◽

pp. 3321-3328 ◽

Cited By ~ 5

Author(s):

Yoshio Okada ◽

Satoshi Tsuboi

Keyword(s):

Amino Acids ◽

Amino Acid ◽

Amino Acid Sequence ◽

Total Synthesis ◽

Human Leukocyte ◽

Cathepsin G ◽

Leukocyte Elastase ◽

Human Leukocyte Elastase ◽

Eglin C ◽

The Relationship

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Amino acids and peptides. XXX. Synthesis of eglin c(41-49) and eglin c(60-63) and examination of their inhibitory activity towards human leukocyte elastase, cathepsin G, porcine pancreatic elastase and .ALPHA.-chymotrypsin.

Chemical and Pharmaceutical Bulletin ◽

10.1248/cpb.39.184 ◽

1991 ◽

Vol 39 (1) ◽

pp. 184-186 ◽

Cited By ~ 2

Author(s):

Satoshi TSUBOI ◽

Miho TAKEDA ◽

Yoshio OKADA ◽

Yoko NAGAMATSU ◽

Junichiro YAMAMOTO

Keyword(s):

Amino Acids ◽

Inhibitory Activity ◽

Human Leukocyte ◽

Cathepsin G ◽

Leukocyte Elastase ◽

Pancreatic Elastase ◽

Human Leukocyte Elastase ◽

Eglin C ◽

Porcine Pancreatic Elastase

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Synthesis of a trihexacontapeptide corresponding to the sequence 8-70 of eglin c and studies on the relationship between the structure and the inhibitory activity against human leukocyte elastase, cathepsin G and α-chymotrypsin

FEBS Letters ◽

10.1016/0014-5793(90)80461-q ◽

1990 ◽

Vol 272 (1-2) ◽

pp. 113-116 ◽

Cited By ~ 8

Author(s):

Yoshio Okada ◽

Satoshi Tsuboi ◽

Yuko Tsuda ◽

Yoko Nagamatsu ◽

Junichiro Yamamoto

Keyword(s):

Inhibitory Activity ◽

Human Leukocyte ◽

Cathepsin G ◽

Leukocyte Elastase ◽

Human Leukocyte Elastase ◽

Eglin C ◽

The Relationship

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Binding of the Recombinant Proteinase Inhibitor Eglin C from LeechHzrudo Medzcznalzsto Human Leukocyte Elastase, Bovine α-Chymotrypsin and Subtilisin Carlsberg: Thermodynamic Study

Journal of Enzyme Inhibition ◽

10.3109/14756368809040723 ◽

1988 ◽

Vol 2 (3) ◽

pp. 167-172 ◽

Cited By ~ 22

Author(s):

Paolo Ascenzi ◽

Gino Amiconi ◽

Enea Menegatti ◽

Mario Guarneri ◽

Martino Bolognesi ◽

...

Keyword(s):

Proteinase Inhibitor ◽

Human Leukocyte ◽

Thermodynamic Study ◽

Leukocyte Elastase ◽

Subtilisin Carlsberg ◽

Human Leukocyte Elastase ◽

Eglin C

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Amino acids and peptides. XXVIII. Synthesis of peptide fragments related to eglin c and studies on the relationship between their structure and effects on human leukocyte elastase, cathepsin G and .ALPHA.-chymotrypsin.

Chemical and Pharmaceutical Bulletin ◽

10.1248/cpb.38.2369 ◽

1990 ◽

Vol 38 (9) ◽

pp. 2369-2376 ◽

Cited By ~ 4

Author(s):

Satoshi TSUBOI ◽

Kazunori NAKABAYASHI ◽

Yoshikazu MATSUMOTO ◽

Naoki TENO ◽

Yuko TSUDA ◽

...

Keyword(s):

Amino Acids ◽

Human Leukocyte ◽

Cathepsin G ◽

Peptide Fragments ◽

Leukocyte Elastase ◽

Human Leukocyte Elastase ◽

Eglin C ◽

The Relationship

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Synthesis of peptide fragments related to eglin c and examination of their inhibitory effect on human leukocyte elastase, cathepsin G and α-chymotrypsin

Biochemical and Biophysical Research Communications ◽

10.1016/0006-291x(89)91591-x ◽

1989 ◽

Vol 161 (1) ◽

pp. 272-275 ◽

Cited By ~ 13

Author(s):

Y. Okada ◽

S. Tsuboi ◽

Y. Tsuda ◽

K. Nakabayashi ◽

Y. Nagamatsu ◽

...

Keyword(s):

Human Leukocyte ◽

Inhibitory Effect ◽

Cathepsin G ◽

Peptide Fragments ◽

Leukocyte Elastase ◽

Human Leukocyte Elastase ◽

Eglin C

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Design, Synthesis, and Enzymatic Evaluation ofN1-Acyloxyalkyl- andN1-Oxazolidin-2,4-dion-5-yl-Substituted β-lactams as Novel Inhibitors of Human Leukocyte Elastase

Journal of Medicinal Chemistry ◽

10.1021/jm0501331 ◽

2005 ◽

Vol 48 (15) ◽

pp. 4861-4870 ◽

Cited By ~ 25

Author(s):

Rui Moreira ◽

Ana Bela Santana ◽

Jim Iley ◽

João Neres ◽

Kenneth T. Douglas ◽

...

Keyword(s):

Human Leukocyte ◽

Leukocyte Elastase ◽

Design Synthesis ◽

Human Leukocyte Elastase

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ChemInform Abstract: FR901451, a Novel Inhibitor of Human Leukocyte Elastase from Flexibacter sp. Part 2. Pharmacological Effect of FR901451.

ChemInform ◽

10.1002/chin.199523247 ◽

2010 ◽

Vol 26 (23) ◽

pp. no-no

Author(s):

T. FUJITA ◽

Y. SHINGUH ◽

A. YAMAZAKI ◽

K. NAKAHARA ◽

M. OKAMOTO ◽

...

Keyword(s):

Human Leukocyte ◽

Pharmacological Effect ◽

Leukocyte Elastase ◽

Human Leukocyte Elastase

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Versatile Multidimensional Chromatographic System for Drug Discovery as Exemplified by the Analysis of a Nonpeptidic Inhibitor of Human Leukocyte Elastase

Journal of Liquid Chromatography &amp Related Technologies ◽

10.1080/10826079608014035 ◽

1996 ◽

Vol 19 (15) ◽

pp. 2527-2540

Author(s):

Roger A. Earley ◽

Leonard P. Tini

Keyword(s):

Drug Discovery ◽

Human Leukocyte ◽

Chromatographic System ◽

Leukocyte Elastase ◽

Human Leukocyte Elastase

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