WITHDRAWN: Design, synthesis and biological evaluation of 3-substituted-4-anilinequinoline as EGFR tyrosine kinase inhibitors

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2012.10.030 ◽

2012 ◽

Author(s):

Yongjun Mao ◽

Kai Xie ◽

Wenxiu Zhu ◽

Jianfeng Li ◽

Hua Xie ◽

...

Keyword(s):

Tyrosine Kinase ◽

Tyrosine Kinase Inhibitors ◽

Kinase Inhibitors ◽

Biological Evaluation ◽

Design Synthesis ◽

Egfr Tyrosine Kinase ◽

Egfr Tyrosine Kinase Inhibitors ◽

Synthesis And Biological Evaluation

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Design, synthesis and biological evaluation of novel pyrimidine, 3-cyanopyridine and m-amino-N-phenylbenzamide based monocyclic EGFR tyrosine kinase inhibitors

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2013.03.053 ◽

2013 ◽

Vol 21 (11) ◽

pp. 3090-3104 ◽

Author(s):

Yongjun Mao ◽

Wenxiu Zhu ◽

Xiaoguang Kong ◽

Zhen Wang ◽

Hua Xie ◽

...

Keyword(s):

Tyrosine Kinase ◽

Tyrosine Kinase Inhibitors ◽

Kinase Inhibitors ◽

Biological Evaluation ◽

Design Synthesis ◽

Egfr Tyrosine Kinase ◽

Egfr Tyrosine Kinase Inhibitors ◽

Synthesis And Biological Evaluation

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Design, Synthesis and Biological Evaluation of Quinoxalin-2(1H)-one Derivatives as EGFR Tyrosine Kinase Inhibitors

Anti-Cancer Agents in Medicinal Chemistry ◽

10.2174/187152061502150116173357 ◽

2015 ◽

Vol 15 (2) ◽

pp. 267-273 ◽

Author(s):

Xuemei Qin ◽

Xiao Han ◽

Liming Hu ◽

Zhipeng Li ◽

Zhufeng Geng ◽

...

Keyword(s):

Tyrosine Kinase ◽

Tyrosine Kinase Inhibitors ◽

Kinase Inhibitors ◽

Biological Evaluation ◽

Design Synthesis ◽

Egfr Tyrosine Kinase ◽

Egfr Tyrosine Kinase Inhibitors ◽

Synthesis And Biological Evaluation

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Synthesis and biological evaluation of irreversible EGFR tyrosine kinase inhibitors containing pyrido[3,4-d]pyrimidine scaffold

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2018.05.039 ◽

2018 ◽

Vol 26 (12) ◽

pp. 3619-3633 ◽

Author(s):

Hao Zhang ◽

Jin Wang ◽

Hong-Yi Zhao ◽

Xue-Yan Yang ◽

Hao Lei ◽

...

Keyword(s):

Tyrosine Kinase ◽

Tyrosine Kinase Inhibitors ◽

Kinase Inhibitors ◽

Biological Evaluation ◽

Egfr Tyrosine Kinase ◽

Egfr Tyrosine Kinase Inhibitors ◽

Synthesis And Biological Evaluation

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Synthesis and Biological Evaluation of Bis(methoxymethyl)-7,8-dihydro-[1,4]dioxino[2,3-g]quinazolines as EGFR Tyrosine Kinase Inhibitors.

10.1002/chin.200607168 ◽

2006 ◽

Vol 37 (7) ◽

Author(s):

Yong Sup Lee ◽

Seon Hee Seo ◽

Beom-Seok Yang ◽

Jae Yeol Lee

Keyword(s):

Tyrosine Kinase ◽

Tyrosine Kinase Inhibitors ◽

Kinase Inhibitors ◽

Biological Evaluation ◽

Egfr Tyrosine Kinase ◽

Egfr Tyrosine Kinase Inhibitors ◽

Synthesis And Biological Evaluation

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Synthesis and Biological Evaluation of Bis(methoxy methyl)-7,8-dihydro-[1,4]dioxino[2,3-g]quinazolines as EGFR Tyrosine Kinase Inhibitors

Archiv der Pharmazie ◽

10.1002/ardp.200500126 ◽

2005 ◽

Vol 338 (10) ◽

pp. 502-505 ◽

Author(s):

Yong Sup Lee ◽

Seon Hee Seo ◽

Beom-Seok Yang ◽

Jae Yeol Lee

Keyword(s):

Tyrosine Kinase ◽

Tyrosine Kinase Inhibitors ◽

Kinase Inhibitors ◽

Biological Evaluation ◽

Egfr Tyrosine Kinase ◽

Egfr Tyrosine Kinase Inhibitors ◽

Synthesis And Biological Evaluation

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The design, synthesis, and biological evaluation of potent receptor tyrosine kinase inhibitors

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2012.06.029 ◽

2012 ◽

Vol 22 (15) ◽

pp. 4979-4985 ◽

Author(s):

Moon H. Kim ◽

Amy Lew Tsuhako ◽

Erick W. Co ◽

Dana T. Aftab ◽

Frauke Bentzien ◽

...

Keyword(s):

Tyrosine Kinase ◽

Tyrosine Kinase Inhibitors ◽

Receptor Tyrosine Kinase ◽

Kinase Inhibitors ◽

Biological Evaluation ◽

Design Synthesis ◽

Synthesis And Biological Evaluation ◽

Receptor Tyrosine Kinase Inhibitors

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Design, Synthesis, and Evaluation of Ribose-Modified Anilinopyrimidine Derivatives as EGFR Tyrosine Kinase Inhibitors

Frontiers in Chemistry ◽

10.3389/fchem.2017.00101 ◽

2017 ◽

Vol 5 ◽

Author(s):

Xiuqin Hu ◽

Disha Wang ◽

Yi Tong ◽

Linjiang Tong ◽

Xia Wang ◽

...

Keyword(s):

Tyrosine Kinase ◽

Tyrosine Kinase Inhibitors ◽

Kinase Inhibitors ◽

Design Synthesis ◽

Egfr Tyrosine Kinase ◽

Egfr Tyrosine Kinase Inhibitors

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Design, synthesis and biological evaluation of substituted pyrrolo[2,3-d]pyrimidines as multiple receptor tyrosine kinase inhibitors and antiangiogenic agents

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2008.04.019 ◽

2008 ◽

Vol 16 (10) ◽

pp. 5514-5528 ◽

Author(s):

Aleem Gangjee ◽

Ojas A. Namjoshi ◽

Jianming Yu ◽

Michael A. Ihnat ◽

Jessica E. Thorpe ◽

...

Keyword(s):

Tyrosine Kinase ◽

Tyrosine Kinase Inhibitors ◽

Receptor Tyrosine Kinase ◽

Kinase Inhibitors ◽

Biological Evaluation ◽

Antiangiogenic Agents ◽

Design Synthesis ◽

Synthesis And Biological Evaluation ◽

Multiple Receptor ◽

Receptor Tyrosine Kinase Inhibitors

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Design, synthesis, and biological evaluation of novel 3-pyrrolo[b]cyclohexylene-2-dihydroindolinone derivatives as potent receptor tyrosine kinase inhibitors

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2013.08.037 ◽

2013 ◽

Vol 23 (20) ◽

pp. 5630-5633 ◽

Author(s):

Lei Ding ◽

Feng Tang ◽

Wei Huang ◽

Qiu Jin ◽

Han Shen ◽

...

Keyword(s):

Tyrosine Kinase ◽

Tyrosine Kinase Inhibitors ◽

Receptor Tyrosine Kinase ◽

Kinase Inhibitors ◽

Biological Evaluation ◽

Design Synthesis ◽

Synthesis And Biological Evaluation ◽

Receptor Tyrosine Kinase Inhibitors

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Part-1: Design, synthesis and biological evaluation of novel bromo-pyrimidine analogs as tyrosine kinase inhibitors

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2016.04.056 ◽

2016 ◽

Vol 119 ◽

pp. 70-82 ◽

Author(s):

Chandrashekar Suradhenupura Munikrishnappa ◽

Sangamesh B. Puranik ◽

G.V. Suresh Kumar ◽

Y. Rajendra Prasad

Keyword(s):

Tyrosine Kinase ◽

Tyrosine Kinase Inhibitors ◽

Kinase Inhibitors ◽

Biological Evaluation ◽

Design Synthesis ◽

Pyrimidine Analogs ◽

Synthesis And Biological Evaluation

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