cyclic prodrugs
Recently Published Documents

TOTAL DOCUMENTS

25
(FIVE YEARS 0)

H-INDEX

11
(FIVE YEARS 0)
Latest Documents Most Cited Documents Contributed Authors Related Sources Related Keywords

Developments in the synthesis of new functionalized bisphosphonate drug candidates such as cyclic prodrugs

2016 ◽  
Vol 191 (11-12) ◽  
pp. 1504-1508 ◽  
Author(s):  
V. A. Pavlov ◽  
F. H. Ebetino ◽  
M. W. Lundy ◽  
J. Joly ◽  
R. L. Dobson ◽  
...  
Keyword(s):  
Drug Candidates ◽  
Cyclic Prodrugs

ChemInform Abstract: Synthesis and Evaluation of Novel Coumarin-Based Esterase-Sensitive Cyclic Prodrugs of Peptidomimetic RGD Analogues with Improved Membrane Permeability.

ChemInform ◽  
2010 ◽  
Vol 30 (30) ◽  
pp. no-no
Author(s):  
Binghe Wang ◽  
Wei Wang ◽  
Gian P. Camenisch ◽  
Jennifer Elmo ◽  
Huijuan Zhang ◽  
...  
Keyword(s):  
Membrane Permeability ◽  
Cyclic Prodrugs

ChemInform Abstract: Synthesis of Coumarin-Based, Esterase-Sensitive Cyclic Prodrugs of Opioid Peptides with Enhanced Membrane Permeability and Enzymic Stability

ChemInform ◽  
2010 ◽  
Vol 31 (32) ◽  
pp. no-no
Author(s):  
Binghe Wang ◽  
Daxian Shan ◽  
Wei Wang ◽  
Huijuan Zhang ◽  
Olafur Gudmundsson ◽  
...  
Keyword(s):  
Membrane Permeability ◽  
Opioid Peptides ◽  
Cyclic Prodrugs

A comparison of the effects of p-glycoprotein inhibitors on the blood–brain barrier permeation of cyclic prodrugs of an opioid peptide (DADLE)

2009 ◽  
Vol 98 (6) ◽  
pp. 2227-2236 ◽  
Author(s):  
Hui Ouyang ◽  
Thomas E. Andersen ◽  
Weiqing Chen ◽  
Rebecca Nofsinger ◽  
Bente Steffansen ◽  
...  
Keyword(s):  
Blood Brain Barrier ◽  
Opioid Peptide ◽  
Brain Barrier ◽  
P Glycoprotein ◽  
Blood Brain ◽  
Cyclic Prodrugs ◽  
Glycoprotein Inhibitors

Factors that restrict intestinal cell permeation of cyclic prodrugs of an opioid peptide (DADLE): Part II. Role of metabolic enzymes in the intestinal mucosa

2009 ◽  
Vol 98 (1) ◽  
pp. 349-361 ◽  
Author(s):  
Hui Ouyang ◽  
Weiqing Chen ◽  
Thomas E. Andersen ◽  
Bente Steffansen ◽  
Ronald T. Borchardt ◽  
...  
Keyword(s):  
Intestinal Mucosa ◽  
Metabolic Enzymes ◽  
Opioid Peptide ◽  
Intestinal Cell ◽  
Cyclic Prodrugs

Effects of Amino Acid Chirality and the Chemical Linker on the Cell Permeation Characteristics of Cyclic Prodrugs of Opioid Peptides

2006 ◽  
Vol 49 (4) ◽  
pp. 1261-1270 ◽  
Author(s):  
Bianca M. Liederer ◽  
Tarra Fuchs ◽  
David Vander Velde ◽  
Teruna J. Siahaan ◽  
Ronald T. Borchardt
Keyword(s):  
Amino Acid ◽  
Opioid Peptides ◽  
Cyclic Prodrugs
Load More ...
Sign in / Sign up

Export Citation Format

Share Document